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Table 1 In vitro pharmacological characteristics of DAT1 variants.

From: The variable number of tandem repeats element in DAT1 regulates in vitro dopamine transporter density

 

hDAT

hDAT Zero

hDAT 9

hDAT 10

Bmax (± S.E.M)

7747 (± 360)

5913 (± 308)

3021 (± 286)

4669 (± 480)

Kd (± S.E.M)

5.44 (± 0.55)

7.77 (± 0.41)

4.98 (± 0.20)

6.69 (± 0.57)

Ki (± S.E.M)

24.77 (± 1.14)

29.13 (± 1.81)

25.00 (± 0.10)

33.39 (± 4.15)